Bioactivity:

SB 243213 dihydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor).

CAS nr:

1780372-25-9

Purity:

98%

Molecular Weight:

501,33

SMILES:

O=C(N1CCC2=C1C=C(C(F)(F)F)C(C)=C2)NC3=CC=C(OC4=CC=CN=C4C)N=C3.[H]Cl.[H]Cl

Formula:

C22H21Cl2F3N4O2

Pathway:

GPCR/G Protein,Neuroscience

Target:

5-HT Receptor,5-HT Receptor