Bioactivity:

AR antagonist 1 is a potent antagonist of the androgen receptor. It binds to E3 ligase ligands with weak binding affinities to VHL protein in the synthesis of PROTAC ARD-266.

CAS nr:

1818885-54-9

Purity:

98%

Molecular Weight:

278,78

SMILES:

N#CC1=CC=C(O[C@H]2C(C)(C)[C@H](N)C2(C)C)C=C1Cl

Formula:

C15H19ClN2O

Pathway:

Endocrinology/Hormones

Target:

Androgen Receptor