Bioactivity:

Autotaxin-IN-1 is a potent autotaxin inhibitor, which has favorable potency (IC50=2.2 nM), PK properties, and a robust PK/PD relationship and it is used in treatment of osteoarthritis pain[1].

CAS nr:

1619971-30-0

Purity:

98%

Molecular Weight:

405,45

SMILES:

O=C(N1CC2=NC(NC3CC4=C(C=CC=C4)C3)=NC=C2C1)COCCC5=CN=NN5

Formula:

C21H23N7O2

Pathway:

Metabolism

Target:

PDE