Bioactivity:

MZP-55 is a selective BRD3/4 degrader based on PROTAC technology(Brd4BD2 with Kd of 8 nM)

CAS nr:

2010159-48-3

Purity:

98%

Molecular Weight:

1080,72

SMILES:

CC(N=CS1)=C1C2=CC=C(CNC([C@@H]3C[C@@H](O)CN3C([C@H](C(C)(C)C)NC(COCCOCCOCCOCCNC(C(C=C4)=CC=C4C5=CC6=C(C=C5)N(C(C)=O)[C@@H](C)C[C@H]6NC7=CC=C(Cl)C=C7)=O)=O)=O)=O)C=C2

Formula:

C57H70ClN7O10S

Pathway:

Chromatin/Epigenetic

Target:

Epigenetic Reader Domain