Bioactivity:

TPC-144 is a potent and selective LSD1 inhibitor with a reversible inhibition mechanism. TPC-144 has antitumor activity in several human AML and SCLC cell lines and xenograft models.

CAS nr:

2098621-17-9

Purity:

98%

Molecular Weight:

515,6

SMILES:

N[C@H]1C[C@H]2CC[C@H](N2C(C3=CC(C4=CC=C(C#N)C(F)=C4)=C(C5=CC=C(CC(C)(O)C)C=C5F)C=C3)=O)C1

Formula:

C31H31F2N3O2

Pathway:

Target: