WZ-3146 T6733
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
WZ3146 is a mutant-selective irreversible inhibitor of EGFR(L858R) and EGFR(E746_A750) with IC50 of 2 nM and 2 nM; does not inhibit ERBB2 phosphorylation (T798I).
CAS nr:
1214265-56-1
Purity:
98%
Molecular Weight:
464,95
SMILES:
CN1CCN(CC1)c1ccc(Nc2ncc(Cl)c(Oc3cccc(NC(=O)C=C)c3)n2)cc1
Formula:
C24H25ClN6O2
Pathway:
Tyrosine Kinase/Adaptors,Angiogenesis,JAK/STAT signaling
Target:
EGFR,EGFR,EGFR
