Bioactivity:

Sepimostat exhibits neuroprotective activity via NR2B N-methyl-D-aspartate receptor antagonism at the Ifenprodil-binding site of the NR2B subunit. Sepimostat dimethanesulfonate inhibits the Ifenprodil binding with a Ki value of 27.7_ﾵM.

CAS nr:

103926-64-3

Purity:

98%

Molecular Weight:

373,41

SMILES:

C1CN=C(N1)NC2=CC=C(C=C2)C(=O)OC3=CC4=C(C=C3)C=C(C=C4)C(=N)N

Formula:

C21H19N5O2

Pathway:

Membrane transporter/Ion channel,Neuroscience

Target:

iGluR,iGluR