Bioactivity:

GS-626510 is an orally bioavailable inhibitor of BET family bromodomains (Kd: 0.59-3.2 nM for BRD2/3/4; IC50: 83 nM and 78 nM for BD1 and BD2).

CAS nr:

1637770-13-8

Purity:

98%

Molecular Weight:

394,47

SMILES:

CC1=C(C2=CC(C3=C4C=CC=NC4=CC=C3C)=C5NC(C6CC6)=NC5=C2)C(C)=NO1

Formula:

C25H22N4O

Pathway:

Chromatin/Epigenetic

Target:

Epigenetic Reader Domain