GeA-69 T5399
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
GeA-69 (GeA69) is a selective and allosteric PARP14 macrodomain 2 (MD2) inhibitor (Kd: 0.86 _M in ITC assays).
CAS nr:
2143475-98-1
Purity:
98%
Molecular Weight:
300,36
SMILES:
CC(=O)Nc1ccccc1-c1cccc2c3ccccc3[nH]c12
Formula:
C20H16N2O
Pathway:
DNA Damage/DNA Repair,Chromatin/Epigenetic
Target:
PARP,PARP
