Bioactivity:

Corticotropin-releasing factor binding protein (CRFBP) inhibitor peptide; displaces CRF from CRFBP. Suppresses body weight gain and increases motor activity in obese rats in vivo.

CAS nr:

TP2047L

Purity:

98%

Molecular Weight:

3220,68

SMILES:

CC[C@@]([H])([C@@]([H])(C(O)=N[C@@](CO)(C(O)=N[C@@](CC(C)([H])C)(C(O)=N[C@@](CC(O)=O)(C(O)=N[C@@](CC(C)([H])C)(C(O)=N[C@](C(O)=N[C@@](CC1=CC=CC=C1)(C(O)=N[C@@](CC2=CN=CN2)(C(O)=N[C@@](CC(C)([H])C)(C(O)=N[C@@](CC(C)([H])C)(C(O)=N[C@@](CCCNC(N)=N)(C(O)=N[C@@](CCC(O)=O)(C(O)=N[C@](C(O)=N[C@@](CC(C)([H])C)(C(O)=N[C@@](CCC(O)=O)(C(O)=N[C@@](CCSC)(C(O)=N[C@]([H])(C(O)=N[C@@](CCCNC(N)=N)(C(O)=N[C@]([H])(C(O)=N[C@@](CCC(O)=O)(C(O)=N[C@@](CCC(O)=N)(C(O)=N[C@@](CC(C)([H])C)(C(O)=N[C@]([H])(C(O)=N[C@@](CCC(O)=N)(C(O)=N[C@@](CCC(O)=N)(C(O)=N[C@]([H])(C(O)=N[C@@](CC3=CN=CN3)(C(O)=N[C@@](CO)(C(O)=O)[H])[H])C)[H])[H])C)[H])[H])[H])C)[H])C)[H])[H])[H])(C(C)([H])C)[H])[H])[H])[H])[H])[H])[H])([C@@](O)([H])C)[H])[H])[H])[H])[H])N)C.CC(O)=O

Formula:

C141H231N41O43S

Pathway:

GPCR/G Protein

Target:

CRFR