Bioactivity:

MZP-54 is a selective degrader of BRD3/4 based on PROTAC technology(Kd of 4 nM for Brd4BD2)

CAS nr:

2010159-47-2

Purity:

98%

Molecular Weight:

1036,67

SMILES:

O=C(NCCOCCOCCOCC(N[C@@H](C(C)(C)C)C(N1C[C@H](O)C[C@H]1C(NCC2=CC=C(C3=C(C)N=CS3)C=C2)=O)=O)=O)C(C=C4)=CC=C4C5=CC6=C(C=C5)N(C(C)=O)[C@@H](C)C[C@H]6NC7=CC=C(Cl)C=C7

Formula:

C55H66ClN7O9S

Pathway:

Chromatin/Epigenetic

Target:

Epigenetic Reader Domain