Bioactivity:

MP-A08 is a highly selective ATP competitive inhibitor of sphingosine kinase (SPHK1) that targets both SphK1 and SphK2 (Ki: 6.9 ﾱ 0.8 _M and 27 ﾱ 3 _M, respectively).

CAS nr:

219832-49-2

Purity:

98%

Molecular Weight:

519,64

SMILES:

O=S(C1=CC=C(C)C=C1)(NC2=CC=CC=C2/C=N/C3=CC=CC=C3NS(=O)(C4=CC=C(C)C=C4)=O)=O

Formula:

C27H25N3O4S2

Pathway:

GPCR/G Protein

Target:

S1P Receptor