Bioactivity:

CMP8 is a selective ligand for estrogen receptor. CMP8 binds to the mutant estrogen receptor ligand binding domain (ERLBD). CMP8 has IC50 values of 29 nM , 41 nM, 1100 nM and 2200 nM for MGER_, MGRER_, hER_ and hER_, respectively.

CAS nr:

851107-28-3

Purity:

98%

Molecular Weight:

528,08

SMILES:

O=C1CCC2(CC3=CC=C(Cl)C=C3)CC4=C(C=CC(O)=C4)C2=C1C5=CC=C(OCCN6CCCCC6)C=C5

Formula:

C33H34ClNO3

Pathway:

Endocrinology/Hormones,Endocrinology/Hormones

Target:

Estrogen Receptor/ERR,Estrogen/progestogen Receptor