CPI-169 racemate T6809
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
CPI-169 is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively.
CAS nr:
1450655-76-1
Purity:
98%
Molecular Weight:
528,66
SMILES:
CCS(=O)(=O)N1CCC(CC1)C(C)n1c2ccccc2c(C(=O)NCc2c(OC)cc(C)[nH]c2=O)c1C
Formula:
C27H36N4O5S
Pathway:
Chromatin/Epigenetic,Chromatin/Epigenetic
Target:
Epigenetic Reader Domain,Histone Methyltransferase
