Bioactivity:

Mardepodect hydrochloride can cross the blood-brain barrier. Mardepodect hydrochloride is an effective and selective PDE10A inhibitor (IC50: 0.37 nM). It has >1000-fold selectivity over other PDEs.

CAS nr:

T16498

Purity:

98%

Molecular Weight:

428,91

SMILES:

CN1N=C(C2=CC=C(OCC3=NC4=CC=CC=C4C=C3)C=C2)C(C5=CC=NC=C5)=C1.Cl[H]

Formula:

C25H21ClN4O

Pathway:

Metabolism

Target:

PDE