Empesertib T8487
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
Empesertib is an orally bioavailable and selective inhibitor Mps1(IC50 < 1 nM), with potential antineoplastic activity.
CAS nr:
1443763-60-7
Purity:
98%
Molecular Weight:
559,61
SMILES:
COc1cc(ccc1Nc1nc2ccc(cn2n1)-c1ccc(NC(=O)[C@H](C)c2ccc(F)cc2)cc1)S(C)(=O)=O
Formula:
C29H26FN5O4S
Pathway:
Cytoskeletal Signaling
Target:
Kinesin
