Bioactivity:

GSK9311 hydrochloride, a less active analog of GSK6853, can be used as a negative control. GSK9311 hydrochloride inhibits BRPF bromodomain (pIC50s: 6.0 and 4.3 for BRPF1 and BRPF2).

CAS nr:

2253733-09-2

Purity:

98%

Molecular Weight:

474

SMILES:

[H]Cl.C[C@@H]1CNCCN1C2=C(N(CC)C(C3=CC=CC=C3OC)=O)C=C(C(N4C)=C2)N(C)C4=O

Formula:

C24H32ClN5O3

Pathway:

Chromatin/Epigenetic

Target:

Epigenetic Reader Domain