Bioactivity:

T-0201 (TA 0201) is a highly potent, long-acting, orally active, and selective ETA receptor antagonist. T-0201 also inhibited ET-1-induced pulmonary artery contraction in isolated rabbits.

CAS nr:

169679-53-2

Purity:

98%

Molecular Weight:

614,52

SMILES:

CC(CO)(C)C1=CC=C(S(NC2=NC=NC(OCCOC3=NC=C(Br)C=N3)=C2C4=CC=C(C)C=C4)(=O)=O)C=C1

Formula:

C27H28BrN5O5S

Pathway:

Target: