Bioactivity:

MK-3207 is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM, highly selective versus human AM1, AM2, CTR, and AMY3. Phase 2.

CAS nr:

957116-20-0

Purity:

98%

Molecular Weight:

594,05

SMILES:

C1CCC2(C1)C(=O)N([C@@H](CN2)C3=CC(=CC(=C3)F)F)CC(=O)NC4=CC5=C(C[C@@]6(C5)C7=C(NC6=O)N=CC=C7)C=C4.Cl

Formula:

C31H29F2N5O3�HCl

Pathway:

Membrane transporter/Ion channel

Target:

CGRP Receptor