Bioactivity:

P300/CBP-IN-5 is a potent inhibitor of p300/CBP histone acetyltransferase (IC50 of 18.8 nM).

CAS nr:

1889284-33-6

Purity:

98%

Molecular Weight:

618,55

SMILES:

O=C(CN(C1=O)C(N[C@@]21C[C@H](C3=C2C=CC(C4=CN(N=C4)CC(NC)=O)=C3)F)=O)N([C@H](C(F)(F)F)C)CC5=CC=C(C=C5)F

Formula:

C29H27F5N6O4

Pathway:

Chromatin/Epigenetic

Target:

Epigenetic Reader Domain